產(chǎn)品詳情
簡(jiǎn)單介紹:
EZH2Inhibitor,EPZ005687
詳情介紹:
Purpose | A potent EZH2 inhibitor |
Characteristics | A potent and selective inhibitor of histone lysine N-methyltransferase EZH2 (Ki = 24 nM). It displays more than 500-fold selectivity against 15 other protein methyltransferases and has 50-fold selectivity against the closely related enzyme, EZH1. |
Purity | ≥ 99?%HPLC |
Chemical Name | 1-Cyclopentyl-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-6-(4-(morpholinomethyl)phenyl)-1H-indazole-4-carboxamide |
Formula | C??H??N?O? |
Permeability | Not-permeable |
Solubility | DMSO |
Molecular Weight | 539.67 g/mol |
CAS-No | 1396772-26-1 |
Restrictions | For Research Use only |
Format | Solid |
Handling Advice | Protect from air and light |
Storage | -20 °C |
Expiry Date | 36 months |
Supplier Images |
|